Copper-mediated C-H(sp2)/C-H(sp3) coupling of benzoic acid derivatives with ethyl cyanoacetate:an ex

来源 :2015年全国药物化学学术会议暨第五届中英药物化学学术会议 | 被引量 : 0次 | 上传用户：battichen

【摘要】

：

An expedient,copper-mediated,direct C-H(sp2)/C-H(sp3)bond coupling of benzoic acid derivatives with ethyl cyanoacetate by the deployment of an 8-aminoquinoline moiety as a bidentate directing group is

【作者】

：

Wei Zhu Dengyou Zhang Nan Yang Hong Liu

【机构】

：

CAS Key Laboratory of Receptor Research,Shanghai Institute of Materia Medica,Chinese Academy of Scie

【出处】

：

2015年全国药物化学学术会议暨第五届中英药物化学学术会议

【发表日期】

：

2015年3期

【关键词】

：

C-H activation copper isoquinolinone ethyl cyanoacetate

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