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,Expression and purification of lipoprotein-associated phospholipase A2, a key enzyme involved in at
[期刊论文] 作者:Fu-jun ZHANG,Mao-jun CAI,Jing-kang SHEN,Yi-ping WANG,
来源:中国药理学报(英文版) 年份:2006
Aim: To express and purify lipoprotein-associated phospholipase A2 (Lp-PLA2), and to establish a screening model for Lp-PLA2 inhibitors using the expressed Lp-P...
[期刊论文] 作者:Dan-qi CHEN,Xin WANG,Lin CHEN,Jin-xue HE,Ze-hong MIAO,Jing-kang SHEN,
来源:中国药理学报(英文版) 年份:2011
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,Identification of non-peptidic neuromedin U receptor modulators by a robust homogeneous screening a
[期刊论文] 作者:Tao MENG,Hao-ran SU,Christoph BINKERT,Walter FISCHLI,Ling ZHOU,Jing-kang SHEN,Ming-wei WANG,
来源:中国药理学报(英文版) 年份:2008
Aim:To develop a homogeneous binding assay for high-throughput screening (HTS) of hit compounds at human neuromedin U receptor (hNMU-R) 1 and to identify non-pe...
[期刊论文] 作者:Jun-lan YU,Tian-tian CHEN,Chen ZHOU,Fu-lin LIAN,Xu-long TANG,Yi WEN,Jing-kang SHEN,
来源:中国药理学报(英文版) 年份:2016
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,Design, synthesis, and anti-inflammatory evaluation of a series of novel amino acid-binding 1,5-dia
[期刊论文] 作者:Ming-hui LI,Lin-lin YIN,Mao-jun CAI,Wei-yu ZHANG,Yue HUANG,Xin WANG,Xing-zu ZHU,Jing-kang SHEN,
来源:中国药理学报(英文版) 年份:2005
Aim: To design and synthesize a series of novel amino acid-binding 1,5-diarylpyrazole derivatives, which are intended to act as prodrugs with better aqueous sol...
Pharmacophore-based design,synthesis,and biological evaluation of novel 3-((3,4-dichlorophenyl)(4-su
[期刊论文] 作者:Dong-Mei Zhao,Wen-Yan Li,Yu-Fang Shi,Xu-Qiong Xiong,Shuai Song,Chen-Zhou Hao,Mao-Sheng Cheng,Jing-Kang Shen,
来源:Chinese Chemical Letters 年份:2014
Cholesteryl ester transfer protein(CETP) is a plasma glycoprotein that plays an important role in decreasing high-density lipoprotein cholesterol(HDL-C) levels...
Construction of a small peptide library related to inhibitor OM99-2 and its structure-activity relat
[期刊论文] 作者:Bin HU,Bing XIONG,Bei-ying QIU,Xin LI,Hai-ping YU,Kun XIAO,Xin WANG,Jia LI,Jing-kang SHEN,
来源:中国药理学报(英文版) 年份:2006
Aim: To develop probes for detecting the binding specificity between β-secretase and substrate, and provide reliable biological activity data for further resea...
[期刊论文] 作者:Shuai CHEN,Li-li CHEN,Hai-bin LUO,Tao SUN,Jing CHEN,Fei YE,Jian-hua CAI,Jing-kang SHEN,Xu SHEN,Hua-liang,
来源:中国药理学报(英文版) 年份:2005
Aim: To characterize enzymatic activity of severe acute respiratory syndrome(SARS) coronavirus (CoV) 3C-like protease (3CLpro) and its four site-directed mutant...
[期刊论文] 作者:Qian CHAI,Yuan-yuan LI,Qiang SHEN,Lan-ping MA,Li-na ZHANG,Xin WANG,Li SHENG,Jing-ya LI,Jia LI,Jing-kang SHEN,
来源:中国药理学报(英文版) 年份:2010
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