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目前,正在研究开发的新的抗结核药有下列几种类型:利福平类药物 (1)KRM-1648(benzox-azinorifamycin):它是新合成的利福平衍生物。动物实验证明,该药对结核菌有抗菌活性;在巨噬细胞内对结核菌有杀菌作用。它在血清内的浓度比利福平稍
Currently, there are the following new types of anti-TB drugs under research and development: Rifampicin (1) Benzoxazinifamycin (KRM-1648): It is a newly synthesized rifampicin derivative. Animal experiments show that the drug has antibacterial activity against Mycobacterium tuberculosis; bactericidal effect on TB in macrophages. Its concentration in serum is slightly less than rifampicin