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报道了用９９ｍＴｃ标记Ｔｅｂｏｒｏｘｉｍｅ（简称ＴＥＢＯ），并在标记后对其质量进行了鉴定。结果表明，其物理性质、化学性质及生物学性质均符合国家制定的放射性药物的质量标准；动物实验表明，小鼠注射量为成人用量的１００倍、观察１５天后，实验组和对照组无差别；注入量为０．１ｍｌ（２０７．ＺｋＢｑ／只），２ｍｉｎ后心肌摄取达峰值１７．７５±０．３３％（ｇｏｒｇａｎ）－１；心肌清除也快，１５ｍｉｎ已清除至８．４２±４．７２％（ｇｏｒｇａｎ）－１。肝脏高峰值在１０ｍｉｎ左右，兔体内的药物动力学特征为快速短时间内完成多体位心肌显像提供药代学基础。
Reported the use of 99mTc labeled Teboroxime (abbreviated TEBO), and its quality was identified after labeling. The results showed that its physical, chemical and biological properties are in line with the national standards for the quality of radiopharmaceuticals; animal experiments show that the amount of mice injected 100 times the amount of adult observation 15 days after the experimental group and the control group no difference ; Injection volume was 0.1ml (207.ZkBq / only), 2 minutes after myocardial uptake of 17.75 ± 0.33% (gorgan) -1; myocardial clearance is also fast, 15min has been cleared to 8.42 ± 4. 72% (gorgan) -1. Liver peak value of about 10min, the pharmacokinetic characteristics of the rabbit in vivo for quick and short multi-body myocardial imaging to provide pharmacokinetic basis.