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雷帕霉素rapamycin(RPM、Rapa)是链霉菌属丝状菌(streptomyces hygro scopicus)发酵产生的一种具有抗真菌作用的大环内脂类抗生素。1975年Vezina和Sehgal从加拿大Rapa Nui岛的土壤中分离出来而得名。1977年Martel等报道其具有免疫抑制作用。1989年Morris等率先将Rapa用于抗移植
Rapamycin rapamycin (RPM, Rapa) is an antifungal macrolide antibiotic produced by the fermentation of Streptomyces hygro scopicus. Vezina and Sehgal got their name from the soil of Rapa Nui Island in Canada in 1975. In 1977, Martel et al reported that they have immunosuppressive effects. In 1989, Morris took the lead in using Rapa for anti-transplantation