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绿十字和旭硝子公司的强效降压药绿十字(GreenCross)和旭硝子(AsahiGlass)公司协作合成了2个可供口服的血管紧张素Ⅱ拮抗剂GA-0050和GA0056.临床前数据提示,它们可能具有潜在的抗高血压作用。这两个化合物作用于Ⅰ型受体,GA-...
Two cross-linked angiotensin II antagonists, GA-0050 and GA0056, were synthesized by Green Cross and Asahi Glass in cooperation with Asahi Glass’s potent antihypertensive drug Green Cross. Preclinical data suggest that they may have potential antihypertensive effects. These two compounds act on type I receptors, GA -...