An NHC-catalyzed assembly of spirocyclic oxindole-cyclopentene

来源 :中国化学会第十三届全国有机合成化学学术研讨会 | 被引量 : 0次 | 上传用户：urgeboy1

【摘要】

：

【作者】

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Jiang Ligen Que Yonglei Li Tuanjie Yu Chenxia Yao Changsheng

【机构】

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School of Chemistry and Chemical Engineering, Jiangsu Key Laboratory of Green Synthetic Chemistry fo

【出处】

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中国化学会第十三届全国有机合成化学学术研讨会

【发表日期】

：

2016年8期

【关键词】

：

N-Heterocyclic Carbene spirocyclic oxindole-cylopentene

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　　The spirocyclic oxindole-cylopentene skeletons featured in a large number of nature products have potential biological activity.Therefore,various approaches such as phosphine catalysis,and metal-mediated multistep transformations,have been performed to realize the successful assembly of spirocyclopentaneoxindole.However,the lengthiness of synthetic route and complexity of the starting materials necessitate the developement of new telescoped protocol to construct this framework.

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An NHC-catalyzed assembly of spirocyclic oxindole-cyclopentene

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