Since the preparation of the first transition metal guanidinate by Lapperts group in 19701,guanidinato([RNC(NR′2)NR]-,R,R′ = alkyl,aryl,silyl,etc)ligands
A series of hybrids from phenylsulfonylfuroxan and anilinopyrimidine were synthesized and biologically evaluated as EGFR inhibitors for intervention of NSCL